產(chǎn)品屬性：
產(chǎn)品名稱 | THIP |
規(guī)格 | 1mg、5mg |
貨號 | EY-01Y14176 |
Cas No.: 64603-91-4
別名: N/A
化學(xué)名: N/A
分子式: C6H8N2O2
分子量: 140.14
溶解度: Soluble in DMSO
儲存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述：
THIP (Gaboxadol) is a selective δ-aminobutyric acid type A receptor (δ-GABAAR) agonist, functionally selective GABAAR ligand, exhibits agonism at α4β1δ, α4β3δ and weak antagonism at αβγ and α4β2δ GABAARs[1].
α4β3δ GABAAR|13 μM (EC50)
[1]. Hoestgaard-Jensen K, et al. Probing α4βδ GABAA receptor heterogeneity: differential regional effects of a functionally selective α4β1δ/α4β3δ receptor agonist on tonic and phasic inhibition in rat brain. J Neurosci. 2014 Dec 3;34(49):16256-72.
特別提醒公司產(chǎn)品僅供科研使用
